IL-1 down-regulates platelet-derived growth factor-alpha receptor gene expression at the transcriptional level in human osteoblastic cells .

Xie JF ; Stroumza J ; Graves DT

Department of Oral Biology , Boston University School of Graduate Dentistry , MA .

J Immunol 153 : 378-83 ( 1994)

Abstract
Regulation of the platelet-derived growth factor ( PDGF)-alpha receptor is thought to play an important role in pathophysiologic processes . Previously , we have reported that IL-1 has the potential to regulate PDGF-induced biologic activity in both normal human osteoblastic cells and the human osteoblastic cell line , MG-63 , by decreasing the expression of PDGF-alpha receptor mRNA . In the present studies , we analyzed the effects of IL-1 on transcription rates and the stability of PDGF-alpha receptor mRNA in MG-63 cells . The data indicate that the t1/2 of PDGF-alpha receptor mRNA is approximately 3.3 h after incubation with the RNA II polymerase transcription inhibitor 5,6-dichloro-1 beta-D-ribofuranosylbenzimidazole ( DRB ) . Approximately the same t1/2 ( 3.1 h ) was obtained when osteoblastic cells were incubated with IL-1 . The t1/2 for PDGF-alpha receptor mRNA for cells incubated with both IL-1 and DRB was 3 h . This finding suggests that the levels of PDGF-alpha receptor mRNA transcripts are not regulated by post-transcriptional mechanisms . Results of nuclear run-on analysis were consistent with this conclusion , demonstrating that IL-1 modulates PDGF-alpha receptor gene expression at the transcriptional level . Surprisingly , incubation of cells with cycloheximide also caused down-regulation of PDGF-alpha receptor mRNA , which suggests that synthesis of a labile factor is necessary for constitutive expression . The functional consequence of down-regulation of PDGF-alpha receptors by IL-1 was also assessed . By using chemotaxis assays , we demonstrated that IL-1 significantly inhibited PDGF-AA-mediated migration in human MG-63 osteoblastic sarcoma cells .